RE: Competition between fibrinogen and PAC-1

From: Kenneth Ault (AULTK@MAIL.MMC.ORG)
Date: Wed Jan 07 1998 - 09:24:54 EST


   I am not an expert in the use of PAC-1, but I think there has been
some misinformation on the list about it and I would like to put in my 2
cents.

PAC-1 is an IgM monoclonal that binds to an epitope of GPIIb/IIIa which
appears upon activation.  The appearance of the epitope requires that
GPIIb/IIIa be in its normal configuration and thus requires the presence
of calcium.  One cannot successfully use PAC-1 on platelets that have
been treated with EDTA (citrate is OK), or with fixed platelets
(fixation seems to induce artifactual binding of PAC-1 to both resting
and activated platelets).

The epitope recognized by PAC-1 is not the fibrinogen binding site.  As
far as I know, there should be no competition between PAC-1 and
fibrinogen.  Other monoclonals, such as 7E3 do recognize the fibrinogen
binding site and will compete with fibrinogen, but I don't think that is
true of PAC-1.

I hope this is helpful.

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Kenneth A. Ault M.D.
Maine Medical Center Research Institute
125 John Roberts Road
Suite #8
South Portland ME 04106

Voice: (207) 761-9090
Fax:    (207) 761-2130
E-Mail:   aultk@mail.mmc.org
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